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Design, Synthesis and in vitro Controlled Release of New Adamantanodiarylketone Antimycobacterials

Publications associées (27)

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A critically degenerate elliptic Dirichlet problem, spectral theory and bifurcation

Charles Stuart

In an open, bounded subset Omega of R-N such that 0 is an element of Omega we consider the nonlinear eigenvalue problem -Sigma(N)(i,j,=1) partial derivative(i){A(ij)(x)partial derivative(j)u} + V(x)u + n(x,del u)+ g(x, u) = lambda u in Omega integral(Omega ...

2020

On the choice of metric in gradient-based theories of brain function

Wulfram Gerstner, Johanni Michael Brea, Jean-Pascal Théodor Pfister

The idea that the brain functions so as to minimize certain costs pervades theoretical neuroscience. Because a cost function by itself does not predict how the brain finds its minima, additional assumptions about the optimization method need to be made to ...

2020

Optimal Spline Generators for Derivative Sampling

Michaël Unser, Shayan Aziznejad, Alireza Naderi

The goal of derivative sampling is to reconstruct a signal from the samples of the function and of its first-order derivative. In this paper, we consider this problem over a shift-invariant reconstruction subspace generated by two compact-support functions ...

IEEE2019

In vitro Controlled Release from Solid Pharmaceutical Formulations of two new Adamantane Aminoethers with Antitubercular Activity (I)

Stewart Cole, Anthony Vocat

The aim of the present investigation was to develop matrix tablet formulations for the in vitro controlled release of 2 new tuberculocidal adamantane aminoethers (compounds I and II), congeneric to the adamantane derivative SQ109 , which is in final clinic ...

Georg Thieme Verlag Kg2017

Contributions to Modelling Extremes of Spatial Data

Linda Frossard

The increasing interest in using statistical extreme value theory to analyse environmental data is mainly driven by the large impact extreme events can have. A difficulty with spatial data is that most existing inference methods for asymptotically justifie ...

EPFL2017

Noether Theorems and Quantum Anomalies

Tudor Ratiu

A quantum anomaly is the breaking of symmetry with respect to some transformations after the quantization of a classical Hamiltonian or Lagrangian system. It is shown that both the Noether theorems (including their infinite-dimensional versions) and the ex ...

Springer Verlag2017

Benzothiophene, benzyloxybenzylidene and indoline derivatives useful for the treatment of tuberculosis

Stewart Cole, Jan Lars Rybniker

The present invention relates to benzothiophene, benzyloxybenzylidene and indoline-2-one derivatives and the use of said derivatives in the treatment and/or prevention of tuberculosis. ...

2016

2-homopiperazine-1-yl-4h-1,3-benzothiazine-4-one derivatives and process for the preparation of 2- (homo)piperazine 1,3-benzothiazine-4-one hydrochlorides

2-homopiperazine-1-yl-4H-l, 3 -bensothiazine-4-one derivatives of formula (I) are provided. They are useful in the treatment of bacterial infections, in particular tuberculosis, buruli ulcer and leprosy. A process for the preparation of 2- (homo)piperazine ...

2016

Bifurcation without Frechet differentiability at the trivial solution

Charles Stuart

Criteria for the bifurcation of small solutions of an equation F(lambda,u) = 0 from a line {(lambda,0): lambda is an element of R} of trivial solutions are usually based on properties of the DuF(lambda,0) at the trivial solutions, where the partial derivat ...

Wiley-Blackwell2015

Discontinuous Galerkin method for fractional convection-diffusion equations

Jan Sickmann Hesthaven

We propose a discontinuous Galerkin method for convection-subdiffusion equations with a fractional operator of order alpha [1,2] defined through the fractional Laplacian. The fractional operator of order alpha is expressed as a composite of first order der ...

Society for Industrial and Applied Mathematics2014

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A critically degenerate elliptic Dirichlet problem, spectral theory and bifurcation

Charles Stuart

2020

On the choice of metric in gradient-based theories of brain function

Wulfram Gerstner, Johanni Michael Brea, Jean-Pascal Théodor Pfister

2020

In vitro Controlled Release from Solid Pharmaceutical Formulations of two new Adamantane Aminoethers with Antitubercular Activity (I)

Stewart Cole, Anthony Vocat

Georg Thieme Verlag Kg2017

2016

2-homopiperazine-1-yl-4h-1,3-benzothiazine-4-one derivatives and process for the preparation of 2- (homo)piperazine 1,3-benzothiazine-4-one hydrochlorides

2016