Concept
Receptor antagonist
Related lectures (36)
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Pharmacodynamics: Ligand Concentration, Binding, and Effect
Explores the relationship between ligand concentration, binding, and effect, focusing on allosteric modulators and types of pharmacological antagonists.
Neurotransmitter Glutamate: Receptor Dynamics and Pharmacodynamics
Explores neurotransmitter dynamics, receptor interactions, and pharmacological concepts in CNS synapses.
Interrogating SAR: Medicinal Chemistry
Covers medicinal chemistry basics, high-throughput screening, lead discovery milestones, and compound selectivity in drug optimization.
Receptor-Ligand Interaction: Quantification and Mechanisms
Explores methods to quantify receptor-ligand interactions, ligand-gated ion channels, and the Hill equation.
Interrogating SAR in Medical Chemistry
Delves into the fundamentals of medicinal chemistry, emphasizing the interrogation of Structure-Activity Relationships (SAR) in drug design.
Receptors and Targeting
Explores receptors, ligands, and their role in signal transduction, including the activation of the immune system and the significance of multivalency in receptor-ligand interactions.
Pharmacodynamics: Ligand-Receptor Binding Kinetics
Explores ligand-receptor binding kinetics, concentration-effect relationship, and drug therapy impact.
Chemical Biology meets Drug Discovery
Explores Chemical Biology, Drug Discovery, enzyme kinetics, and inhibition methods, including competitive and non-competitive inhibition.
Inhibitor Design & Analysis
Covers the design and analysis of inhibitors for next-generation covalent drugs, focusing on target engagement and the importance of cysteine targeting.