An efficient procedure for the regioselective monoprotection of 1,2-diols

Jieping Zhu
1992
Article

Résumé

Regioselective nucleophilic ring opening of isopropylidene ketals of simple diols or sugars, e.g. I (R = Ac, CH2Ph), by AlMe3 gave the corresponding II (R = H, CH2PH). This reagent offers a new method for selective monoprotection of 1,2-diols. [on SciFinder (R)]

Source officielle

https://infoscience.epfl.ch/record/158215?ln=fr

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