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Lecture
Pharmacokinetics: Drug Absorption and Distribution
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Identifying Correct Target in Medical Chemistry
Explores target identification, efficacy, and safety in medical chemistry, emphasizing the importance of on-target specificity and drug design.
Pharmacokinetic & Pharmacodynamic Evaluations
Covers the principles of pharmacokinetics and pharmacodynamics, including drug exposure-response relationships.
Interrogating Drugs' Mode of Action
Delves into enzyme inhibition, reversible and irreversible binding, and covalent drugs, exploring drug modes of action and their impact on drug efficacy.
Pharmacokinetic & Pharmacodynamic Studies
Discusses the importance of assessing PK/PD relationships in drug development and the use of multiple PD biomarkers.
Drug Targets: Adrenergic Signaling
Explores drug targets and adrenergic signaling, covering receptors, enzymes, and transporter proteins.
Drug Metabolism: Xenobiotics and Enzymes
Explores drug metabolism, focusing on xenobiotics, enzymes, biotransformation reactions, and factors affecting drug metabolism.
Selective Drug Targeting Mechanisms
Explores selective drug targeting mechanisms, resistance development, tuberculosis incidence, BCR-ABL mutations, tyrosine kinase inhibitors, drug toxicity, interactions, and toxicology studies.
Pharmacokinetics Modeling: Zero and First-Order Kinetics
Explores pharmacokinetics modeling, covering zero and first-order kinetics, drug distribution, and key parameters for drug elimination.
Pharmacological Targets and Interventions
Explores targets for drug action and the design of specific inhibitors.
Pharmacodynamics: Acid-sensing ion channels and Drug Targets
Explores acid-sensing ion channels, drug targets, and ligand-receptor binding.